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Synthesis and proteasome inhibition of N-allyl vinyl ester-based peptides
Baldisserotto, Anna; Franceschini, Christian; Scalambra, Franco; Trapella, Claudio; Marastoni, Mauro; Sforza, Fabio; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
JOURNAL OF PEPTIDE SCIENCE
Vol. 16, No. 11, pp: 659-663, Anno: 2010

α,β-Unsaturated N-Acylpyrrole Peptidyl Derivatives: New Proteasome Inhibitors
Baldisserotto, Anna; Ferretti, Valeria; Destro, Federica; Franceschini, Christian; Marastoni, Mauro; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 53, No. 17, pp: 6511-6515, Anno: 2010

New cyclic peptide proteasome inhibitors
Baldisserotto, Anna; Marastoni, Mauro; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 19, No. 7, pp: 1966-1969, Anno: 2009

N-Terminal-prolonged vinyl ester-based peptides as selective proteasome b1 subunit inhibitors
Baldisserotto, Anna; Destro, Federica; Vertuani, Gianni; Marastoni, Mauro; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY
Vol. 17, No. 15, pp: 5535-5540, Anno: 2009

Structure-activity relationship study of position 4 in the urotensin-II receptor ligand U-II(4-11)
Marzola, Erika; Camarda, Valeria; Batuwangala, Madura Suharshana; Lamberti, Dg; Calo', Girolamo; Guerrini, Remo; Trapella, Claudio; Regoli, Domenico; Tomatis, Roberto; Salvadori, Severo     dettagli >>
Elsevier Science Incorporated / NY Journals:Madison Square Station, PO Box 882:New York, NY 10159:(212)633-3730, EMAIL: usinfo-f@elsevier.com, INTERNET: http://www.elsevier.com, Fax: (212)633-3680, PEPTIDES
Vol. 29, No. 5, pp: 674-679, Anno: 2008

Vinyl ester-based cyclic peptide proteasome inhibitors
Baldisserotto, Anna; Marastoni, Mauro; Fiorini, Stella; Pretto, Loretta; Ferretti, Valeria; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 18, No. 6, pp: 1849-1854, Anno: 2008

Peptide-based molecules for the production of positive charged liposomes and micelles
Cortesi, Rita; Marastoni, Mauro; Tomatis, Roberto; Menegatti, Enea; Esposito, Elisabetta; Nastruzzi, Claudio     dettagli >>
JOURNAL OF MICROENCAPSULATION
Vol. 25, No. 2, pp: 71-81, Anno: 2008

C-terminal constrained phenylalanine as a pharmacophoric unit in peptide-based proteasome inhibitors
Baldisserotto, Anna; Marastoni, Mauro; Lazzari, Ilaria; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664, EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 43, No. 7, pp: 1403-1411, Anno: 2008

Glutamine vinyl ester proteasome inhibitors selective for trypsin-like (beta2) subunit
Baldisserotto, Anna; Marastoni, Mauro; Trapella, Claudio; Gavioli, Riccardo; Ferretti, Valeria; Pretto, Loretta; Tomatis, Roberto     dettagli >>
Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664, EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 42, No. 5, pp: 586-592, Anno: 2007

P3 and P4 position analysis of vinyl ester pseudopeptide proteasome inhibitors
Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 16, No. 12, pp: 3125-3130, Anno: 2006

Synthesis and biological evaluation of new vinyl ester pseudotripeptide proteasome inhibitors
Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 41, No. 8, pp: 978-984, Anno: 2006

HIV protease inhibitors: synthesis and activity of N-aryl-N '-hydroxyalkyl hydrazide pseudopeptides
Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Mcdonald, J; Bortolotti, Fabrizio; Tomatis, Roberto     dettagli >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 40, No. 1, pp: 445-451, Anno: 2005

Peptidyl vinyl ester derivatives: New class of selective inhibitors of proteasome trypsin-like activity
Marastoni, Mauro; Baldisserotto, Anna; Cellini, Silvia; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 48, No. 15, pp: 5038-5042, Anno: 2005

Proteasome inhibitors: synthesis and activity of arecoline oxide tripeptide derivatives
Marastoni, Mauro; Mcdonald, J.; Baldisserotto, Anna; Canella, Alessandro; DE RISI, Carmela; Pollini, Gian Piero; Tomatis, Roberto     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 14, No. 1, pp: 1965-1968, Anno: 2004

Arecoline tripeptide inhibitors of proteasome
Marastoni, Mauro; Baldisserotto, Anna; Canella, Alessandro; Gavioli, Riccardo; DE RISI, Carmela; Pollini, Gian Piero; Tomatis, Roberto     dettagli >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 47, No. 6, pp: 1587-1590, Anno: 2004

Cytotoxic T lymphocyte epitope analogues containing cis- or trans-4-aminocyclohexanecarboxylic acid residues
Marastoni, M.; Bazzaro, M.; Micheletti, F.; Gavioli, R.; Tomatis, R.     dettagli >>
BIOORGANIC & MEDICINAL CHEMISTRY
Vol. 10, No. 9, pp: 3061-3066, Anno: 2002

Effect of interferon-alpha therapy on epitope-specific cytotoxic T lymphocyte responses in hepatitis C virus-infected individuals
Vertuani, S; Bazzaro, M; Gualandi, G; Micheletti, F; Marastoni, Mauro; Fortini, Cinzia; Canella, Alessandro; Marino, M; Tomatis, Roberto; Traniello, Maria Serena; Gavioli, Riccardo     dettagli >>
EUROPEAN JOURNAL OF IMMUNOLOGY
Vol. 32, No. 1, pp: 144-154, Anno: 2002

Peptide analogues of a subdominant epitope expressed in EBV-associated tumors: synthesis and immunological activity
Marastoni, Mauro; Bazzaro, M.; Micheletti, F.; Gavioli, Riccardo; Tomatis, Roberto     dettagli >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 44, No. 14, pp: 2370-2373, Anno: 2001

Further studies on nociceptin-related peptides: Discovery of a new chemical template with antagonist activity on the nociceptin receptor
Guerrini, Remo; Calo', Girolamo; Bigoni, R; Rizzi, Anna; Varani, Katia; Toth, G; Gessi, Stefania; Hashiba, E; Hashimoto, Y; Lambert, Dg; Borea, Pier Andrea; Tomatis, Roberto; Salvadori, Severo; Regoli, Domenico     dettagli >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 43, No. 1, pp: 2805-2813, Anno: 2000

A CD4/T4 receptor peptide ligand labeled with technetium-99m: Synthesis and biological activity
Boschi, Alessandra; Uccelli, Licia; Bolzati, Cristina; Marastoni, Mauro; Tomatis, Roberto; Spisani, Susanna; Traniello, Maria Serena; Piffanelli, Adriano     dettagli >>
NUCLEAR MEDICINE AND BIOLOGY
Vol. 27, No. 8, pp: 791-795, Anno: 2000

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